SCHEMBL9708697

SCHEMBL9708697

CCCn1c(=O)c2c(nc(C(C)C)n2Cc2ccc(-c3ccccc3)c(-c3nnn[nH]3)c2)n(-c2ccccc2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 11/20 0.39
ADORA1 P30542 3/20 0.39
ADORA2B P29275 4/20 0.36
ADORA2A P29274 3/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708757 0.92 ADORA3 (0.41) ADORA3ADORA1ADORA2BADORA2A
SCHEMBL9707680 0.91 ADORA3 (0.43) ADORA3ADORA1ADORA2BADORA2AKDM4E
SCHEMBL9707906 0.88 AGTR1 (0.38) ADORA3ADORA1ADORA2AKMT2A
SCHEMBL9707425 0.86 ADORA3 (0.41) ADORA3ADORA1ADORA2BADORA2A
SCHEMBL9707898 0.85 MAPT (0.38) ADORA3ADORA1KMT2A
SCHEMBL9708047 0.84 USP1 (0.39) ADORA3KDM4EMEN1ALDH1A1KMT2A
SCHEMBL9707739 0.84 ADORA3 (0.47) ADORA3ADORA1ADORA2BADORA2A
SCHEMBL9707519 0.84 ADORA3 (0.39) ADORA3ADORA1ADORA2BADORA2AKMT2A
SCHEMBL9708310 0.84 RAB9A (0.42) ADORA3ADORA1ADORA2BADORA2AMEN1
SCHEMBL9708591 0.84 ADORA1 (0.40) ADORA3ADORA1ADORA2BADORA2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed