SCHEMBL9708640

SCHEMBL9708640

COCCn1c(=O)[nH]c2nc(C(C)C)n(Cc3ccc(-c4ccccc4-c4nnn[nH]4)cc3)c2c1=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
USP1 O94782 11/20 0.42
PKM P14618 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
DCTPP1 Q9H773 1/20 0.37
PPARG P37231 1/20 0.36
GAA P10253 1/20 0.36
RECQL P46063 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TSHR P16473 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708424 0.91 ADORA2B (0.40) USP1PPARG
SCHEMBL9708226 0.90 AGTR1 (0.38) USP1PPARG
SCHEMBL9708519 0.90 DCTPP1 (0.42) USP1PKMKDM4EALDH1A1DCTPP1
SCHEMBL9708314 0.89 ADORA2B (0.38) USP1PPARG
SCHEMBL9707736 0.89 ADORA3 (0.42) USP1PPARG
SCHEMBL9707407 0.88 GPR18 (0.39) USP1KDM4EPPARG
SCHEMBL9707560 0.88 PPARG (0.42) USP1PPARGKMT2A
SCHEMBL9707572 0.88 AGTR1 (0.41) PKMKDM4EALDH1A1DCTPP1PPARG
SCHEMBL9707717 0.87 ALDH1A1 (0.49) USP1PKMKDM4EALDH1A1GAA
SCHEMBL9708637 0.87 PPARG (0.37) USP1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed