SCHEMBL9709861

SCHEMBL9709861

Cc1cc(NCc2ccc(-c3ccccc3C(=O)OC(C)(C)C)cc2)c2ncccc2n1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 12/20 0.47
AGTR1 P30556 1/20 0.43
AGTR2 P50052 1/20 0.43
CD38 P28907 3/20 0.41
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709560 0.87 CD38 (0.50) AGTR1AGTR2CD38
SCHEMBL27791830 0.78 CYP2C19 (0.47) CD38
SCHEMBL9494718 0.77 ACP1 (0.54) BDKRB1AGTR1AGTR2CD38
SCHEMBL9709862 0.76 BDKRB1 (0.46) BDKRB1AGTR1AGTR2
SCHEMBL9709569 0.75 PPARG (0.48) BDKRB1AGTR1AGTR2ADRA1A
SCHEMBL9377391 0.75 MAPT (0.48) BDKRB1
SCHEMBL3058636 0.74 CD38 (0.56) BDKRB1CD38
SCHEMBL9709799 0.74 CD38 (0.47) BDKRB1AGTR1AGTR2CD38
SCHEMBL9709866 0.73 AGTR1 (0.47) AGTR1AGTR2
Hydrochloric Acid SCHEMBL9494706 0.73 CD38 (0.55) BDKRB1CD38

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO disclosed