SCHEMBL9713845

SCHEMBL9713845

CN(C)c1ccc(S(=O)(=O)c2ccc(N)cc2)c(N(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.46
ALDH1A1 P00352 3/20 0.46
CYP3A4 P08684 2/20 0.46
ALOX15 P16050 2/20 0.46
TP53 P04637 1/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
LMNA P02545 1/20 0.46
MPO P05164 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PKM P14618 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HKDC1 Q2TB90 1/20 0.39
HSD11B1 P28845 1/20 0.37
CA12 O43570 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713990 0.89 HTR6 (0.50) HTR6ALDH1A1CYP3A4TDP1LMNA
SCHEMBL9713635 0.84 ALDH1A1 (0.46) HTR6ALDH1A1CYP3A4ALOX15TP53
SCHEMBL9713941 0.80 ALDH1A1 (0.46) HTR6ALDH1A1CYP3A4ALOX15TDP1
SCHEMBL17774674 0.79 HTR6 (0.50) HTR6ALDH1A1CYP3A4TDP1LMNA
SCHEMBL9713804 0.77 GAA (0.53) ALDH1A1LMNATSHRPKMMEN1
SCHEMBL30543085 0.74 HTR6 (0.53) HTR6ALDH1A1CYP3A4ALOX15TP53
SCHEMBL21378334 0.74 HTR6 (0.53) HTR6ALDH1A1CYP3A4ALOX15TP53
SCHEMBL9713818 0.74 PKM (0.63) ALDH1A1LMNATSHRPKMMEN1
SCHEMBL17774692 0.72 HTR6 (0.46) HTR6ALDH1A1CYP3A4TDP1LMNA
SCHEMBL16638466 0.71 CA12 (0.68) HTR6ALDH1A1CYP3A4ALOX15TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed