SCHEMBL9714155

SCHEMBL9714155

Cc1ncn(Cc2c(F)cccc2F)c1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA5A P35218 1/20 0.47
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
TSHR P16473 2/20 0.37
PKM P14618 2/20 0.37
MAPK1 P28482 1/20 0.37
CD38 P28907 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
C1S P09871 4/20 0.36
KLKB1 P03952 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
AXL P30530 1/20 0.35
FLT3 P36888 1/20 0.35
MERTK Q12866 1/20 0.35
GAA P10253 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714294 0.84 CA5A (0.48) CA5AKDM4EALDH1A1ADORA2AADORA1
SCHEMBL10568675 0.82 ALDH1A1 (0.49) KDM4EALDH1A1TSHRMAPK1MEN1
SCHEMBL9714307 0.82 CA5A (0.46) CA5AKDM4EALDH1A1ADORA2AADORA1
SCHEMBL31333084 0.79 CA5A (0.52) CA5AADORA2AADORA1TSHRMAPK1
SCHEMBL31333042 0.77 CA5A (0.44) CA5ATSHRPKMMAPK1CD38
SCHEMBL18050891 0.76 TSHR (0.47) CA5AKDM4EALDH1A1TSHRPKM
SCHEMBL9714543 0.75 LMNA (0.55) ALDH1A1GAAMEN1KMT2A
SCHEMBL9714280 0.74 CA5A (0.57) CA5AKDM4EALDH1A1PKMCD38
SCHEMBL10571269 0.73 ALDH1A1 (0.48) KDM4EALDH1A1TSHRMEN1KMT2A
SCHEMBL9714161 0.72 CA5A (0.48) CA5AKDM4EALDH1A1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0248414-B1 ARALKYL IMIDAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1992-09-23 EP disclosed
US-4851424-A 1-Phenyl-lower alkyl-imidazole 4- or 5-carboxamide compounds which are useful in the treatment of epilepsy CIBA-GEIGY CORPORATION (US) 1989-07-25 US disclosed
EP-0248414-A2 Aralkyl imidazole derivatives CIBA-GEIGY AG (CH) 1987-12-09 EP disclosed