SCHEMBL9714265

SCHEMBL9714265

CNC(=O)c1cn(Cc2c(F)cccc2F)cn1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.42
CA5A P35218 1/20 0.42
KLKB1 P03952 4/20 0.41
GAA P10253 1/20 0.40
SCD O00767 1/20 0.39
SMYD3 Q9H7B4 1/20 0.39
PDE4A P27815 1/20 0.37
PDE7A Q13946 1/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
JAK3 P52333 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM5B Q9UGL1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714339 0.87 RIPK1 (0.41) RIPK1CA5AKLKB1SCDSMYD3
SCHEMBL9714332 0.87 KLKB1 (0.44) RIPK1CA5AKLKB1SMYD3CYP2C19
SCHEMBL10568102 0.84 MEN1 (0.46) RIPK1CA5AKLKB1SCDJAK2
SCHEMBL12179543 0.83 CA5A (0.46) RIPK1CA5AKLKB1KDM5B
SCHEMBL9714146 0.82 CA5A (0.58) RIPK1CA5AKLKB1JAK2JAK1
SCHEMBL10568262 0.79 ALDH1A1 (0.48) CA5AGAA
SCHEMBL18377475 0.79 KLKB1 (0.56) RIPK1KLKB1SCDCYP2C19KDM5B
SCHEMBL21316959 0.77 PTGS1 (0.53)
SCHEMBL21316963 0.76 POLB (0.41) KLKB1GAACYP2C19
SCHEMBL15838648 0.76 CA5A (0.69) CA5AKLKB1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0248414-B1 ARALKYL IMIDAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1992-09-23 EP claimed
EP-0248414-A2 Aralkyl imidazole derivatives CIBA-GEIGY AG (CH) 1987-12-09 EP claimed
EP-0248414-B1 ARALKYL IMIDAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1992-09-23 EP disclosed
EP-0248414-A2 Aralkyl imidazole derivatives CIBA-GEIGY AG (CH) 1987-12-09 EP disclosed