SCHEMBL9714951

SCHEMBL9714951

CNC(=O)Cc1c(N(C)C)n[nH]c1-c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.39
POLB P06746 1/20 0.39
NPY5R Q15761 1/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
RAB9A P51151 2/20 0.35
MAPT P10636 1/20 0.35
NPC1 O15118 1/20 0.35
NR1I2 O75469 1/20 0.35
AHR P35869 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TSPO P30536 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KDM4E B2RXH2 1/20 0.34
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9715039 0.89 LMNA (0.42) P2RX7POLBRAB9AMAPTSMN1; SMN2
SCHEMBL9715021 0.86 PTGDR2 (0.39) NPY5RRAB9AMAPTNPC1NR1I2
Hydrochloric Acid SCHEMBL9715064 0.85 PTGDR2 (0.39) NPY5RRAB9AMAPTNPC1NR1I2
SCHEMBL9715049 0.81 RAB9A (0.54) POLBRAB9AMAPTSMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL9714965 0.80 RAB9A (0.53) POLBRAB9AMAPTSMN1; SMN2KDM4E
SCHEMBL9715038 0.77 L3MBTL1 (0.43) POLBRAB9ASMN1; SMN2KDM4EPTGS2
Hydrochloric Acid SCHEMBL9714943 0.76 L3MBTL1 (0.45) POLBRAB9ASMN1; SMN2KDM4EPTGS2
Hydrochloric Acid SCHEMBL9714930 0.73 LMNA (0.41) POLBMAPTKDM4E
SCHEMBL8514273 0.68 P2RX7 (0.47) P2RX7POLBRAB9ANPC1SMN1; SMN2
SCHEMBL12809523 0.67 POLB (0.61) POLBRAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5057534-A Anxiolytic, anticonfulsant and muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1991-10-15 US claimed
WO-1992018484-A1 3-AMINO-5-ARYLPYRAZOLE-4-ACETIC ACID DERIVATIVES EXHIBITING THERAPEUTIC EFFECTS A.H. ROBINS COMPANY, INCORPORATED (US) 1992-10-29 WO disclosed
US-5057534-A Anxiolytic, anticonfulsant and muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1991-10-15 US disclosed