SCHEMBL9719043

SCHEMBL9719043

CCCOc1c(OC)cc(CO)cc1SC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HPGD P15428 2/20 0.40
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
MGAM O43451 3/20 0.39
GAA P10253 3/20 0.39
SI P14410 3/20 0.39
MGAM2 Q2M2H8 3/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTGS2 P35354 1/20 0.39
TUBB4A P04350 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9719060 0.88 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2HPGDMEN1HTT
SCHEMBL9719016 0.82 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2HPGDMEN1HTT
SCHEMBL9718999 0.79 HSD17B10 (0.65) HSD17B10ALOX15TSHRALDH1A1SMN1; SMN2
SCHEMBL19632491 0.78 ALOX15 (0.48) HSD17B10ALOX15TSHRSMN1; SMN2PTGS2
SCHEMBL9719068 0.75 ALDH1A1 (0.45) TSHRALDH1A1SMN1; SMN2HPGDMEN1
SCHEMBL9124419 0.75 S1PR2 (0.48)
SCHEMBL9829357 0.74 TUBB4A (0.41) ALDH1A1SMN1; SMN2HPGDMEN1HTT
SCHEMBL9829388 0.74 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2MEN1KMT2AGAA
SCHEMBL2744248 0.74 TSHR (0.50) HSD17B10ALOX15TSHRALDH1A1SMN1; SMN2
SCHEMBL20436811 0.73 S1PR2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132463-A Cardiovascular, skin, kidney, respiratory system, and gastrointestinal disorders MERCK & CO., INC. (US) 1992-07-21 US disclosed
EP-0257921-B1 NEW 1,3-DIARYL CYCLOPENTANES AND DERIVATIVES THEREOF AS PAF ANTAGONISTS MERCK & CO. INC. (US) 1992-04-15 EP disclosed
US-5047420-A Platelet activating factor MERCK & CO., INC. (US) 1991-09-10 US disclosed
EP-0257921-A2 New 1,3-diaryl cyclopentanes and derivatives thereof as paf antagonists MERCK & CO. INC. (US) 1988-03-02 EP disclosed