SCHEMBL9719060

SCHEMBL9719060

CCCOc1c(OC)cc(CCl)cc1SC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HPGD P15428 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
PTGS2 P35354 1/20 0.39
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
TUBB2A Q13885 1/20 0.37
TUBB8 Q3ZCM7 1/20 0.37
TUBA3E Q6PEY2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9719043 0.88 HSD17B10 (0.42) ALDH1A1SMN1; SMN2HPGDMAPTKDM4E
SCHEMBL9719016 0.82 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2HPGDMAPTKDM4E
SCHEMBL9719068 0.75 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2HPGDMAPTKDM4E
SCHEMBL19818498 0.72 PTGS2 (0.67) ALDH1A1SMN1; SMN2HPGDMAPTPTGS2
SCHEMBL9829388 0.71 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2MAPTKDM4ELMNA
SCHEMBL9829357 0.71 TUBB4A (0.41) ALDH1A1SMN1; SMN2HPGDMEN1HTT
SCHEMBL1706883 0.71 PTGS2 (0.64) MAPTKDM4EPTGS2TUBB4ATUBB
SCHEMBL20970860 0.71 HTR2A (0.74) ALDH1A1SMN1; SMN2HPGDMAPTKDM4E
SCHEMBL29633103 0.71 HTR2A (0.74) ALDH1A1SMN1; SMN2HPGDMAPTKDM4E
SCHEMBL14569424 0.70 TTR (0.55) ALDH1A1SMN1; SMN2HPGDMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132463-A Cardiovascular, skin, kidney, respiratory system, and gastrointestinal disorders MERCK & CO., INC. (US) 1992-07-21 US disclosed
EP-0257921-B1 NEW 1,3-DIARYL CYCLOPENTANES AND DERIVATIVES THEREOF AS PAF ANTAGONISTS MERCK & CO. INC. (US) 1992-04-15 EP disclosed
US-5047420-A Platelet activating factor MERCK & CO., INC. (US) 1991-09-10 US disclosed
EP-0257921-A2 New 1,3-diaryl cyclopentanes and derivatives thereof as paf antagonists MERCK & CO. INC. (US) 1988-03-02 EP disclosed