SCHEMBL9720753

SCHEMBL9720753

CN1C(=O)CN(C2CCCCC2N2CC(=O)N(C)C(=O)C2)CC1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.32
APP P05067 1/20 0.32
BACE1 P56817 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
OPRL1 P41146 1/20 0.31
BRD4 O60885 1/20 0.31
BRD2 P25440 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA4 P22748 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA7 P36544 1/20 0.30
CHRNA4 P43681 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720917 1.00 ALDH1A1 (0.37) ALDH1A1LMNAMAPK1APPBACE1
SCHEMBL9720921 1.00 ALDH1A1 (0.37) ALDH1A1LMNAMAPK1APPBACE1
SCHEMBL23660680 0.82 LMNA (0.46) LMNAMAPK1OPRL1GSK3AGSK3B
SCHEMBL8912497 0.68 TSHR (0.35) ALDH1A1LMNAKDM4ETDP1
SCHEMBL13103999 0.68 ALDH1A1 (0.33) ALDH1A1
SCHEMBL8912493 0.68 TSHR (0.35) ALDH1A1LMNAKDM4ETDP1
SCHEMBL9846845 0.68 ALDH1A1 (0.39) ALDH1A1LMNAOPRL1KDM4EHSD17B10
SCHEMBL8914442 0.68 TSHR (0.35) ALDH1A1LMNAKDM4ETDP1
SCHEMBL9846838 0.68 ALDH1A1 (0.39) ALDH1A1LMNAOPRL1KDM4EHSD17B10
SCHEMBL9846852 0.68 ALDH1A1 (0.39) ALDH1A1LMNAOPRL1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992000740-A2 BIS-DIOXOPIPERAZINES AND THEIR USE AS PROTECTION AGENTS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1992-01-23 WO claimed
WO-2021144746-A1 USE OF ICRF-193 DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING THEREOF FOR THE PREVENTION OF CHRONIC CUMULATIVE CARDIOTOXICITY CAUSED BY THERAPY WITH ANTHRACYCLINE ANTICANCER DRUGS UNIVERZITA KARLOVA V PRAZE (CZ) 2021-07-22 WO disclosed
WO-1992000740-A2 BIS-DIOXOPIPERAZINES AND THEIR USE AS PROTECTION AGENTS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1992-01-23 WO disclosed