SCHEMBL9720774

SCHEMBL9720774

COc1ccc(C(CCN2CCN(Cc3ccc(O)cc3)CC2)c2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.60
CCR5 P51681 3/20 0.54
MAPT P10636 2/20 0.54
TDP1 Q9NUW8 1/20 0.54
CCR2 P41597 4/20 0.54
HTR1A P08908 1/20 0.53
KDM4E B2RXH2 1/20 0.52
MAPK1 P28482 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6766190 0.82 CCR2 (0.84) SIGMAR1CCR5CCR2
SCHEMBL9720795 0.81 CCR2 (0.54) SIGMAR1CCR2
SCHEMBL6770892 0.79 CCR2 (0.87) CCR5CCR2
SCHEMBL11848227 0.79 CCR2 (0.73) SIGMAR1CCR2KDM4E
SCHEMBL9720800 0.79 SIGMAR1 (0.56) SIGMAR1MAPK1
Hydrochloric Acid SCHEMBL11838606 0.77 CCR2 (0.71) SIGMAR1CCR2KDM4E
SCHEMBL28217942 0.77 SIGMAR1 (1.00) SIGMAR1KDM4E
SCHEMBL8963508 0.77 HTR1A (0.53) SIGMAR1CCR5MAPTTDP1HTR1A
SCHEMBL11842606 0.77 CCR5 (0.60) SIGMAR1CCR5KDM4EMAPK1
SCHEMBL25326051 0.76 SIGMAR1 (0.64) SIGMAR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5142052-A Cationic effect-driven carbinol/amine reaction LABORATOIRES SYNTEX (FR) 1992-08-25 US disclosed