SCHEMBL9723348

SCHEMBL9723348

O=C(O)C[C@H](NC(=O)C(F)(F)F)C(=O)Nc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.46
CASP7 P55210 1/20 0.44
CASP9 P55211 1/20 0.44
CASP6 P55212 1/20 0.44
CASP8 Q14790 1/20 0.44
MMP2 P08253 2/20 0.43
MMP3 P08254 2/20 0.43
GAA P10253 1/20 0.43
POLB P06746 1/20 0.42
PDK1 Q15118 2/20 0.42
PDK2 Q15119 2/20 0.42
PDK3 Q15120 2/20 0.42
PDK4 Q16654 2/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HDAC3 O15379 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14254895 0.79 HDAC1 (0.56) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL7829245 0.75 MAPT (0.49) MMP2MMP3GAAPOLBPDK1
SCHEMBL11566967 0.75 MAPT (0.47) GAAPOLBPDK1PDK2PDK3
SCHEMBL10591792 0.74 ALDH1A1 (0.57) POLBHSD17B10
SCHEMBL9301420 0.74 ALDH1A1 (0.57) POLBHSD17B10
SCHEMBL27183189 0.74 MLYCD (0.44) MMP2GAAHDAC1HDAC7HDAC8
SCHEMBL23080544 0.73 HTT (0.57) GAAPOLBMEN1NPC1TP53
SCHEMBL5611391 0.73 CA2 (0.47) CASP3GAAMAPT
SCHEMBL7832189 0.73 CA2 (0.47) CASP3GAAMAPT
SCHEMBL473070 0.73 CA2 (0.47) CASP3GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5078129-A Therapy for dry mouth RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 1992-01-07 US disclosed
US-4839352-A ANTIBIOTICS MERCK & CO., INC. (US) 1989-06-13 US disclosed
US-4820506-A ALLEVIATING DRY MOUTH OR XEROSTOMIA; MIXTURE OF ORGANIC ACIDS, SWEETENER AND CALCIUM PHOSPHATE RESEARCH FOUNDATION, STATE UNIVERSITY OF NEW YORK (US) 1989-04-11 US disclosed