SCHEMBL9725445

SCHEMBL9725445

COc1ccc2c(c1)[nH]c(=O)n2CCN(C)C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CCR4 P51679 1/20 0.47
HTR2A P28223 2/20 0.46
HTR2C P28335 2/20 0.46
HTR6 P50406 4/20 0.44
DYRK1A Q13627 1/20 0.44
CALCRL Q16602 1/20 0.43
PDE3B Q13370 2/20 0.43
PDE3A Q14432 2/20 0.43
PDE2A O00408 1/20 0.41
HTR1A P08908 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1E P28566 1/20 0.41
HTR7 P34969 1/20 0.41
HTR5A P47898 1/20 0.41
MYLK Q15746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9725523 0.99 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10CCR4
SCHEMBL9725490 0.89 HTR2A (0.49) KDM4EALDH1A1HPGDHSD17B10CCR4
Hydrochloric Acid SCHEMBL9725431 0.88 HTR2A (0.48) KDM4EALDH1A1HPGDHSD17B10CCR4
SCHEMBL9725370 0.82 DAO (0.53) ALDH1A1HPGDCCR4CALCRLPDE3B
Hydrochloric Acid SCHEMBL9725468 0.81 DAO (0.51) ALDH1A1HPGDCCR4CALCRLPDE3B
SCHEMBL9725470 0.81 MPO (0.45) ALDH1A1HPGDCCR4LMNAMPO
SCHEMBL9725479 0.81 CCR4 (0.56) KDM4EALDH1A1HPGDHSD17B10CCR4
SCHEMBL8125879 0.80 KMO (0.55) KDM4EALDH1A1HPGDHSD17B10DYRK1A
SCHEMBL9725397 0.80 ALDH1A1 (0.55) KDM4EALDH1A1HPGDHSD17B10CCR4
Hydrochloric Acid SCHEMBL9725461 0.80 CCR4 (0.55) KDM4EALDH1A1HSD17B10CCR4HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5162318-A Which have pulmonary surfactant secretion promoting activity YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1992-11-10 US disclosed
EP-0454330-A1 Benzimidazolinone derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-10-30 EP disclosed