SCHEMBL9727495

SCHEMBL9727495

COc1ccc(CC2Oc3ccc(O)cc3C2C)cc1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
CALM1 P0DP23 2/20 0.41
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
CYP3A4 P08684 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ESR1 P03372 7/20 0.39
ESR2 Q92731 7/20 0.39
TLR9 Q9NR96 1/20 0.39
CYP26A1 O43174 1/20 0.38
EDNRB P24530 1/20 0.37
EDNRA P25101 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727737 0.76 ESR1 (0.42) CALM1MEN1KMT2AESR1ESR2
SCHEMBL9727632 0.75 DRD2 (0.39) MEN1KMT2AESR1ESR2
SCHEMBL14102710 0.75 ESR1 (0.49) ALDH1A1MEN1KMT2AESR1ESR2
SCHEMBL14102385 0.75 ESR1 (0.49) ALDH1A1MEN1KMT2AESR1ESR2
SCHEMBL18435584 0.71 MIF (0.40) ALDH1A1HPGDKMT2AESR1ESR2
SCHEMBL13899934 0.69 PTGES (0.46) CYP3A4ESR1ESR2
SCHEMBL9132550 0.68 GLA (0.51) ALDH1A1CYP3A4KMT2ASMN1; SMN2TLR9
SCHEMBL4953164 0.66 ALDH1A1 (0.51) ALDH1A1MEN1CYP3A4KMT2AATM
SCHEMBL14534500 0.64 PTGES (0.46) MEN1KMT2AESR1ESR2
SCHEMBL15033096 0.64 ESR1 (0.42) CYP3A4ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed