SCHEMBL9727632

SCHEMBL9727632

COc1ccc(CC2Oc3cc(CCCOc4ccccc4)c(O)cc3C2C)cc1

nearest known ligand 0.73

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
KCNH2 Q12809 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRB2 P07550 1/20 0.37
ESR1 P03372 1/20 0.37
CYP19A1 P11511 1/20 0.37
ESR2 Q92731 1/20 0.37
PPARD Q03181 2/20 0.35
PPARG P37231 1/20 0.35
FFAR1 O14842 1/20 0.35
NR1H3 Q13133 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727672 0.86 ABCB1 (0.43) DRD2
SCHEMBL9727737 0.83 ESR1 (0.42) MEN1KMT2AADRB2ESR1CYP19A1
SCHEMBL9727495 0.75 ALDH1A1 (0.43) MEN1KMT2AESR1ESR2
SCHEMBL9727705 0.71 ABCB1 (0.41) DRD2MEN1KMT2A
SCHEMBL9727477 0.67 MTNR1B (0.37) DRD2DRD4DRD3ESR1CYP19A1
SCHEMBL9854748 0.64 MTNR1A (0.49) DRD2DRD4DRD3KCNH2MEN1
SCHEMBL10459597 0.63 MAOB (0.45) PPARDPPARG
SCHEMBL5287776 0.63 KCNA3 (0.73) DRD2DRD4DRD3KCNH2MEN1
SCHEMBL1171680 0.62 TDP1 (0.69) DRD2DRD4DRD3KCNH2MEN1
SCHEMBL1172476 0.62 TDP1 (0.69) DRD2DRD4DRD3KCNH2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed