SCHEMBL9727737

SCHEMBL9727737

COc1ccc(CC2Oc3cc(CCCCc4ccc(Cl)cc4)c(O)cc3C2C)cc1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.42
CYP19A1 P11511 1/20 0.42
ESR2 Q92731 1/20 0.42
IGF1R P08069 2/20 0.42
ALOX15 P16050 2/20 0.42
CALM1 P0DP23 1/20 0.37
SLC5A2 P31639 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LTB4R Q15722 1/20 0.35
ADRB2 P07550 1/20 0.35
CNR1 P21554 1/20 0.34
FPR2 P25090 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727632 0.83 DRD2 (0.39) ESR1CYP19A1ESR2MEN1KMT2A
SCHEMBL9727495 0.76 ALDH1A1 (0.43) ESR1ESR2CALM1MEN1KMT2A
SCHEMBL9727793 0.69 ESR1 (0.44) ESR1CYP19A1ESR2IGF1RALOX15
SCHEMBL25328659 0.65 ESR1 (0.69) ESR1CYP19A1ESR2IGF1RALOX15
SCHEMBL5253951 0.63 TAAR1 (0.59) CALM1KMT2ACNR1FPR2
SCHEMBL8702849 0.62 IGF1R (0.61) ESR1CYP19A1ESR2IGF1RALOX15
SCHEMBL4254058 0.62 CALM1 (0.72) IGF1RALOX15CALM1L3MBTL1
Broussonin A SCHEMBL774802 0.61 ESR1 (1.00) ESR1CYP19A1ESR2IGF1RALOX15
SCHEMBL5252007 0.61 CALM1 (0.60) IGF1RALOX15CALM1L3MBTL1
SCHEMBL17400406 0.60 CALM1 (0.69) IGF1RALOX15CALM1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed