SCHEMBL9877259

SCHEMBL9877259

Cc1nn2c(-c3ccccc3C(F)(F)F)ccnc2c1C(=O)N=CN(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 10/20 0.43
PIM1 P11309 10/20 0.43
CHEK1 O14757 3/20 0.40
CDK2 P24941 3/20 0.40
CSNK2A1 P68400 3/20 0.40
MAPT P10636 3/20 0.39
THRB P10828 1/20 0.39
ACVR1 Q04771 2/20 0.38
NPC1 O15118 2/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9877170 0.83 NTRK1 (0.64) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL9877172 0.83 NTRK1 (0.64) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL9728870 0.81 NTRK1 (0.65) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL9878320 0.81 KDM4E (0.48) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL9728647 0.81 KDM4E (0.48) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL9728729 0.79 NTRK1 (0.53) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL9877954 0.69 MAPT (0.53) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL9877951 0.69 MAPT (0.53) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL11465849 0.64 BRAF (0.59) MAPTNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL9877207 0.63 KDM4E (0.67)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5059691-A Anxiolytic agents; hypotensive agents; nervous system disorders; cognition activators AMERICAN CYANAMID COMPANY (US) 1991-10-22 US disclosed