SCHEMBL9729621

SCHEMBL9729621

COc1ccc2c(c1)OCCC2CN(O)C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.47
ALOX5 P09917 8/20 0.47
KDM4C Q9H3R0 3/20 0.43
USP2 O75604 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8103275 0.79 HTR1A (0.56) HTR1AKDM4CUSP2CYP3A4
Hydrochloric Acid SCHEMBL8112970 0.77 HTR1A (0.55) HTR1AKDM4CUSP2CYP3A4
SCHEMBL5175120 0.76 HTR1A (0.54) HTR1AKDM4CUSP2CYP3A4
SCHEMBL11000702 0.76 HTR1A (0.43) HTR1AUSP2CYP3A4
SCHEMBL5226604 0.76 MTNR1A (0.61) HTR1AKDM4C
Formamide SCHEMBL9729628 0.75 HTR1A (0.59) HTR1AKDM4CUSP2CYP3A4
SCHEMBL5172931 0.75 HTR1A (0.56) HTR1AKDM4CUSP2CYP3A4
SCHEMBL5223865 0.74 MTNR1A (0.63) HTR1A
SCHEMBL9464927 0.74 HTR1A (0.63) HTR1AKDM4CUSP2CYP3A4
SCHEMBL9695945 0.73 ALOX5 (0.74) ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5155130-A Lipoxygenase inhibitors CIBA-GEIGY CORPORATION (US) 1992-10-13 US disclosed
EP-0412939-A2 Certain benzopyran and benzothiopyran derivatives CIBA-GEIGY AG (CH) 1991-02-13 EP disclosed