SCHEMBL9733215

SCHEMBL9733215

CS(=O)(=O)Nc1ccc2c(c1)C(=O)C(C1CCN(CCc3ccc4nonc4c3)CC1)C2

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.59
KCNJ1 P48048 4/20 0.47
DRD2 P14416 2/20 0.39
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
SIGMAR1 Q99720 1/20 0.39
HTR1A P08908 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
HTR7 P34969 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9807574 0.87 DRD2 (0.47) KCNH2DRD2HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL9592944 0.86 DRD2 (0.46) KCNH2DRD2HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL9731916 0.85 KCNH2 (0.51) KCNH2KCNJ1HTR1AHTR7
Methyl Alcohol SCHEMBL9591993 0.85 DRD2 (0.45) KCNH2DRD2HTR2AHTR2CHTR2B
SCHEMBL9807598 0.79 SIGMAR1 (0.58) DRD2HTR2AHTR2CHTR2BSIGMAR1
Hydrochloric Acid SCHEMBL9591965 0.78 DRD2 (0.57) KCNH2DRD2HTR2AHTR2CHTR2B
SCHEMBL9593272 0.78 ADRA1D (0.57) KCNH2DRD2HTR2AHTR2CHTR2B
SCHEMBL9592174 0.78 ACHE (0.59) DRD2HTR2AHTR1AHTR7
SCHEMBL9732081 0.77 KCNH2 (0.61) KCNH2KCNJ1DRD2HTR2AHTR2C
Hydrochloric Acid SCHEMBL9593896 0.77 ADRA1D (0.56) KCNH2DRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112824-A Benzofurazan compounds MERCK & CO., INC. (US) 1992-05-12 US disclosed