SCHEMBL9733222

SCHEMBL9733222

CC1(C)C=C(n2cc(N)ccc2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.34
BACE1 P56817 11/20 0.32
PGR P06401 2/20 0.32
NSD2 O96028 1/20 0.32
CASP3 P42574 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
CTSD P07339 2/20 0.32
MALT1 Q9UDY8 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
ALK Q9UM73 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733851 0.87 MAOB (0.34) POLBBACE1PGRNSD2CASP3
SCHEMBL9735211 0.87 ABCC9 (0.34) POLBPGRNSD2CASP3MALT1
SCHEMBL9733322 0.84 KCNJ1 (0.36) PGRALDH1A1KMT2AALK
SCHEMBL9735213 0.84 POLB (0.33) POLBBACE1PGRNSD2CASP3
SCHEMBL9733571 0.84 POLB (0.33) POLBBACE1PGRNSD2CASP3
SCHEMBL9733284 0.82 HTR1A (0.37) POLBBACE1PGRNSD2CASP3
SCHEMBL9735233 0.81 PGR (0.36) PGR
SCHEMBL9733957 0.80 CYP19A1 (0.35) POLBBACE1PGRCASP3MALT1
SCHEMBL9734137 0.80 BACE1 (0.35) POLBBACE1PGRNSD2CASP3
SCHEMBL9734001 0.80 POLB (0.33) POLBBACE1PGRNSD2CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed