SCHEMBL9733957

SCHEMBL9733957

CC1(C)C=C(n2cnccc2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.35
ABCC9 O60706 2/20 0.34
CYP11B2 P19099 5/20 0.33
CYP11B1 P15538 1/20 0.33
PGR P06401 2/20 0.32
BACE1 P56817 2/20 0.32
POLB P06746 1/20 0.32
CASP3 P42574 1/20 0.32
MALT1 Q9UDY8 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
GSK3B P49841 2/20 0.31
SRPK2 P78362 1/20 0.31
SRPK1 Q96SB4 1/20 0.31
BUB1 O43683 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9734020 0.83 CYP11B2 (0.37) CYP11B2PGRBACE1POLBCASP3
SCHEMBL9733774 0.83 HTR1A (0.38) CYP19A1ABCC9CYP11B2CYP11B1PGR
SCHEMBL9735211 0.82 ABCC9 (0.34) ABCC9PGRPOLBCASP3MALT1
SCHEMBL9733284 0.82 HTR1A (0.37) ABCC9PGRBACE1POLBCASP3
SCHEMBL9733222 0.80 POLB (0.34) PGRBACE1POLBCASP3MALT1
SCHEMBL9733851 0.80 MAOB (0.34) ABCC9PGRBACE1POLBCASP3
SCHEMBL9733106 0.79 PGR (0.34) CYP11B2CYP11B1PGRBACE1POLB
SCHEMBL9733622 0.79 POLB (0.35) ABCC9PGRBACE1POLBCASP3
SCHEMBL8077234 0.78 PDE4A (0.42) ABCC9CASP3MALT1
SCHEMBL9733784 0.78 CYP11B2 (0.35) ABCC9CYP11B2CYP11B1PGRBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed