SCHEMBL9735211

SCHEMBL9735211

CC1(C)C=C(n2cc(Cl)ccc2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 3/20 0.34
PGR P06401 3/20 0.32
POLB P06746 1/20 0.32
CASP3 P42574 1/20 0.32
CNR2 P34972 1/20 0.32
TP53 P04637 1/20 0.32
MDM2 Q00987 1/20 0.32
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
MALT1 Q9UDY8 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
DRD2 P14416 1/20 0.31
DRD1 P21728 1/20 0.31
KCNH2 Q12809 1/20 0.31
HSD17B3 P37058 1/20 0.31
MIF P14174 2/20 0.31
NSD2 O96028 1/20 0.30
GPR6 P46095 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733851 0.87 MAOB (0.34) ABCC9PGRPOLBCASP3MALT1
SCHEMBL9733222 0.87 POLB (0.34) PGRPOLBCASP3MALT1HTR2A
SCHEMBL9734810 0.86 ABCC9 (0.32) ABCC9PGRPOLBCASP3MALT1
SCHEMBL9734001 0.84 POLB (0.33) ABCC9PGRPOLBCASP3NSD2
SCHEMBL9733322 0.84 KCNJ1 (0.36) ABCC9PGRKCNH2
SCHEMBL9733957 0.82 CYP19A1 (0.35) ABCC9PGRPOLBCASP3MALT1
SCHEMBL9733284 0.82 HTR1A (0.37) ABCC9PGRPOLBCASP3NSD2
SCHEMBL9735233 0.81 PGR (0.36) PGRDRD2
SCHEMBL9733247 0.81 VCAM1 (0.39) ABCC9
SCHEMBL9733571 0.80 POLB (0.33) PGRPOLBCASP3NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed