SCHEMBL9733267

SCHEMBL9733267

CCC1(CC)C=C(n2ccccc2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
PGR P06401 3/20 0.35
BACE1 P56817 3/20 0.32
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3B P49841 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
NSD2 O96028 1/20 0.32
ELANE P08246 1/20 0.32
CASP3 P42574 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733783 0.89 HTR1A (0.36) HTR1AALDH1A1LMNATSHRPGR
SCHEMBL9733284 0.86 HTR1A (0.37) HTR1AALDH1A1PGRBACE1GABRA1
SCHEMBL9733608 0.82 HTR1A (0.36) HTR1AALDH1A1PGRBACE1CCNB2
SCHEMBL9733278 0.81 PGR (0.36) HTR1AALDH1A1PGRBACE1
SCHEMBL9737787 0.79 F10 (0.39) ALDH1A1
SCHEMBL9589614 0.79 ABCC9 (0.38) HTR1APGRGABRA1GABRG2GABRB3
SCHEMBL9733561 0.77 PGR (0.36) HTR1AALDH1A1PGRBACE1NSD2
SCHEMBL8088666 0.77 CASP3 (0.34) HTR1APGRELANECASP3
SCHEMBL8085392 0.76 HTR1A (0.35) HTR1APGR
SCHEMBL9732955 0.75 CYP19A1 (0.44) HTR1AGABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed