SCHEMBL9733908

SCHEMBL9733908

COC(=O)c1ccc2c(c1)C(n1nc(O)ccc1=O)=CC(C)(C)C2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.36
CASP3 P42574 1/20 0.36
PDK2 Q15119 3/20 0.35
BACE1 P56817 1/20 0.35
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TRPA1 O75762 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
XDH P47989 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
PDPK1 O15530 1/20 0.34
AURKA O14965 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9734080 0.81 PDE4B (0.36) OPRM1ALDH1A1TDP1OPRD1MEN1
SCHEMBL10697118 0.79 RAB9A (0.37) CASP3PDK2ALDH1A1SMN1; SMN2ATM
SCHEMBL9733895 0.79 PDK2 (0.39) CASP3PDK2ALDH1A1SMN1; SMN2ATM
SCHEMBL9733491 0.78 CASP3 (0.36) CASP3PDK2ALDH1A1SMN1; SMN2ATM
SCHEMBL9372349 0.71 RAB9A (0.37) OPRM1CASP3ALDH1A1SMN1; SMN2ATM
SCHEMBL8088431 0.71 CNR2 (0.37) OPRM1CASP3ALDH1A1SMN1; SMN2ATM
SCHEMBL9733741 0.68 GABRA1 (0.41) ALDH1A1SMN1; SMN2KDM4ETDP1MEN1
SCHEMBL13131194 0.68 CASP3 (0.44) CASP3PDK2BACE1ALDH1A1SMN1; SMN2
SCHEMBL10697215 0.67 S100A4 (0.34) PDK2KDM4E
SCHEMBL9734695 0.66 KMT2A (0.40) PDK2ALDH1A1TDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed