SCHEMBL9738296

SCHEMBL9738296

O=C(O)Cc1ccc(N2C(=O)CCC23CCC(=O)N3c2ccc(CC(=O)O)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.46
POLB P06746 1/20 0.46
GRK2 P25098 1/20 0.46
CASP6 P55212 1/20 0.46
CTDSP1 Q9GZU7 1/20 0.46
KLKB1 P03952 1/20 0.45
CTSB P07858 1/20 0.45
QPCT Q16769 1/20 0.45
CA2 P00918 1/20 0.42
CAMK2A Q9UQM7 1/20 0.42
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
SRD5A2 P31213 1/20 0.40
AKR1B1 P15121 1/20 0.40
LMNA P02545 2/20 0.40
ABCC4 O15439 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8722675 0.78 ESR1 (0.44) TSHRMMP13
SCHEMBL9730386 0.76 MMP13 (0.59) MMP13MMP2MMP3MMP9
SCHEMBL22184094 0.75 CA12 (0.59) NSD2POLBGRK2CASP6CTDSP1
SCHEMBL10392048 0.74 MMP13 (0.50) GAATSHRMMP13MMP2MMP3
SCHEMBL9644504 0.74 MMP13 (0.35) POLBMMP13MMP2MMP3MMP9
SCHEMBL5124270 0.73 ALDH1A1 (0.66) POLBLMNA
SCHEMBL6788342 0.73 ALDH1A1 (0.61) NSD2POLBGRK2CASP6CTDSP1
SCHEMBL9730839 0.73 MMP13 (0.52) POLBLMNAHTTMMP13MMP2
SCHEMBL6074717 0.69 ITGB3 (0.59) NSD2POLBGRK2CASP6CTDSP1
SCHEMBL9874462 0.69 MMP13 (0.50) POLBLMNAMMP13MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112938-A CYANO- AND CARBOXY-SUBSTITUTED SPIRODILACTAMS SHELL OIL COMPANY (US) 1992-05-12 US disclosed
US-5037948-A Cyano- and carboxy-substituted spirodilactams SHELL OIL COMPANY (US) 1991-08-06 US disclosed