SCHEMBL9739222

SCHEMBL9739222

N#CC1(C#N)OC1c1ccccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.36
PTGS2 P35354 1/20 0.36
MEN1 O00255 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
TP53 P04637 2/20 0.34
RECQL P46063 1/20 0.34
ALDH1A1 P00352 7/20 0.34
MAPT P10636 2/20 0.34
TAAR1 Q96RJ0 1/20 0.34
THRB P10828 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
LMNA P02545 2/20 0.33
TSHR P16473 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
ALOX12 P18054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738560 0.74 ALDH1A1 (0.38) KMT2APTGS2MEN1RECQLALDH1A1
SCHEMBL13802689 0.72 TP53 (0.36) KMT2AMEN1HTR2AHTR2CHTR2B
SCHEMBL10703931 0.72 MAPT (0.42) KMT2APTGS2MEN1ALDH1A1MAPT
SCHEMBL17684053 0.68 OPRL1 (0.40) PTGS2HTR2AHTR2CHTR2BTP53
SCHEMBL11201145 0.65 TSHR (0.47) KMT2APTGS2MEN1HTR2AHTR2C
SCHEMBL9059555 0.65 CHRNB2 (0.36) KMT2AMEN1ALDH1A1HPGD
SCHEMBL17684321 0.65 PTGS2 (0.36) KMT2APTGS2HTR2AHTR2CHTR2B
SCHEMBL17683936 0.63 OPRL1 (0.39) PTGS2HTR2AHTR2CHTR2BTP53
SCHEMBL17683935 0.63 OPRL1 (0.39) PTGS2HTR2AHTR2CHTR2BTP53
SCHEMBL9667454 0.63 PTGS2 (0.35) PTGS2HTR2AHTR2CHTR2BTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082842-A Sedatives HOFFMANN-LA ROCHE INC. (US) 1992-01-21 US disclosed
US-4889854-A MUSCLE RELAXANT, SEDATIVE-HYPNOTIC, ANXIOLYTIC AND-OR ANTICONVULSANT ACTIVITY HOFFMAN-LA ROCHE INC. (US) 1989-12-26 US disclosed
EP-0294599-A2 Tricyclic pyridone derivatives F. HOFFMANN-LA ROCHE AG (CH) 1988-12-14 EP disclosed