SCHEMBL9739396

SCHEMBL9739396

COc1cc(OC)cc(OCCCN2CCCCC2C(C)N2CCc3cc4c(cc3CC2=O)OCO4)c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CYP2D6 P10635 1/20 0.33
DRD2 P14416 1/20 0.33
HRH3 Q9Y5N1 5/20 0.32
KCNH2 Q12809 1/20 0.32
DRD1 P21728 1/20 0.32
EDNRA P25101 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739283 0.85 HRH3 (0.41) HRH3
Hydrochloric Acid SCHEMBL9739083 0.84 HRH3 (0.40) HRH3
SCHEMBL9740494 0.81 SMN1; SMN2 (0.39) MAOAMAOBHRH3KCNH2
SCHEMBL9739398 0.81 MAOA (0.36) MAOAMAOBDRD2HRH3KCNH2
SCHEMBL9740102 0.77 KCNH2 (0.41) CYP2D6HRH3KCNH2
SCHEMBL9740238 0.76 ABCB1 (0.42) HRH3
Hydrochloric Acid SCHEMBL9740197 0.76 CYP3A4 (0.42) HRH3
SCHEMBL9740267 0.75 HRH3 (0.44) HRH3KCNH2
Hydrochloric Acid SCHEMBL9739389 0.75 HRH3 (0.43) HRH3KCNH2
SCHEMBL9740418 0.74 ABCB1 (0.46) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed