SCHEMBL9739556

SCHEMBL9739556

COc1c(Cl)cc2[nH]c[c]c2c1Cl

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHUK O15111 1/20 0.36
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
AKR1B1 P15121 1/20 0.33
DBH P09172 1/20 0.32
TPMT P51580 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
DRD2 P14416 1/20 0.30
DRD1 P21728 1/20 0.30
DRD5 P21918 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6011025 0.75 ALDH1A1 (0.34) ALDH1A1
SCHEMBL9740600 0.74 ALDH1A1 (0.33) ALDH1A1
SCHEMBL4885600 0.74 CSNK2A1 (0.32)
SCHEMBL21614387 0.69 ALDH1A1 (0.42) CHUKAKR1B1TPMTKDM4EALDH1A1
SCHEMBL9740520 0.68 CHUK (0.39) CHUKGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9300156 0.67 ALDH1A1 (0.35) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9739295 0.66 TUBB4A (0.33) KDM4EALDH1A1
SCHEMBL481060 0.65 CYP3A4 (0.50) CHUKAKR1B1TPMTKDM4EALDH1A1
SCHEMBL29749746 0.65 CYP3A4 (0.50) CHUKAKR1B1TPMTKDM4EALDH1A1
SCHEMBL10946322 0.65 GAA (0.48) CHUKTPMTKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed