SCHEMBL9744164

SCHEMBL9744164

O=[C]c1ccccc1CCBr

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.39
PTPN1 P18031 2/20 0.31
GSK3B P49841 2/20 0.31
CYP1A1 P04798 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP1B1 Q16678 1/20 0.31
FFAR1 O14842 1/20 0.31
TAAR1 Q96RJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3021179 0.82 TRPA1 (0.35) CYP1A1CYP1A2CYP1B1
SCHEMBL910448 0.78 DAO (0.38) TDP1CYP1A2FFAR1
SCHEMBL9036603 0.78 TAAR1 (0.50) CYP1A2TAAR1
SCHEMBL5728797 0.78 CYP19A1 (0.43) TDP1CYP1A1CYP1A2CYP1B1FFAR1
SCHEMBL30252315 0.78 CYP19A1 (0.43) TDP1CYP1A1CYP1A2CYP1B1FFAR1
SCHEMBL6210675 0.77 HTR1A (0.44) TDP1FFAR1TAAR1
SCHEMBL30600 0.75 TDP1 (0.55) TDP1PTPN1GSK3BCYP1A1CYP1A2
SCHEMBL2119420 0.75 CYP3A4 (0.44) TDP1CYP1A2
SCHEMBL3822531 0.75 ALDH1A1 (0.35)
SCHEMBL535892 0.75 GABRA1 (0.45) FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101522657-B STAT3/5 activation inhibitor OTSUKA PHARMACEUTICAL CO.,LTD. (JP) 2014-10-15 CN disclosed
CN-1993339-B Aromatic compound OTSUKA PHARMA CO LTD 2013-05-22 CN disclosed
CN-101522657-A STAT3/5 activation inhibitor OTSUKA PHARMA CO LTD (JP) 2009-09-02 CN disclosed
CN-1993339-A Aromatic compound OTSUKA PHARMA CO LTD (JP) 2007-07-04 CN disclosed
CN-1114590-C Unsaturated oximino ether bactericide SHENYAN CHEMICAL ENGINEERING I (CN) 2003-07-16 CN disclosed
CN-1169989-A Process for preparing dithiocarbonimide derivatives SUMITOMO CHEMICAL CO (JP) 1998-01-14 CN disclosed
US-5098996-A Fluorination of compounds for use in diagnosis of nuclear medicine THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1992-03-24 US disclosed