SCHEMBL9746239

SCHEMBL9746239

COC(=O)c1ccc2cc(C(=O)c3ccc4c(c3)C(C)(C)C(C)C4(C)C)ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 2/20 0.48
CYP26A1 O43174 3/20 0.46
RARA P10276 1/20 0.46
RARB P10826 1/20 0.46
RARG P13631 1/20 0.46
CYP26B1 Q9NR63 1/20 0.46
LCK P06239 1/20 0.43
CYP3A4 P08684 3/20 0.41
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
HDAC1 Q13547 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA12 O43570 1/20 0.40
CA7 P43166 1/20 0.40
XDH P47989 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10355823 0.90 CYP3A4 (0.43) CYP26A1RARBRARGCYP3A4ALDH1A1
SCHEMBL9746735 0.85 RARB (0.63) CYP26A1RARARARBRARGCYP26B1
SCHEMBL10544739 0.83 RARB (0.48) CYP26A1RARARARBRARGCYP26B1
SCHEMBL9746813 0.81 RARB (0.43) CYP26A1RARARARBRARGCYP26B1
SCHEMBL9747005 0.80 RARB (0.60) PTPN11CYP26A1RARARARBRARG
SCHEMBL9185753 0.80 CYP3A4 (0.50) CYP26A1CYP3A4ALDH1A1CA1CA2
SCHEMBL9748837 0.78 CYP26B1 (0.46) CYP26A1RARARARBRARGCYP26B1
SCHEMBL9822364 0.77 RARB (0.42) CYP26A1RARARARBRARGCYP26B1
SCHEMBL8522801 0.77 RXRA (0.60) CYP26A1RARARARBRARGCYP26B1
SCHEMBL29365729 0.75 PTPN11 (0.68) PTPN11LCKCYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220118-B1 BICYCLIC NAPHTHALENIC DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN HUMAN AND VETERINARY MEDICINE AND COSMETICS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA - CIRD GALDERMA (FR) 1992-01-02 EP claimed