SCHEMBL9747889

SCHEMBL9747889

CC1C(=O)Nc2c(C(=O)c3ccc(Br)cc3)cccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.44
MAPT P10636 3/20 0.40
NPC1 O15118 3/20 0.40
MAPK1 P28482 2/20 0.40
HTT P42858 2/20 0.40
LMNA P02545 4/20 0.39
ABCB11 O95342 1/20 0.39
PTGS1 P23219 1/20 0.39
ADORA1 P30542 1/20 0.39
PTGS2 P35354 1/20 0.39
KMT2A Q03164 3/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 3/20 0.36
MEN1 O00255 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KDM4E B2RXH2 1/20 0.35
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
CCNB2 O95067 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10949720 0.86 ALDH1A1 (0.34) MAPTLMNAKMT2ARAB9AMEN1
SCHEMBL9748582 0.86 NR4A1 (0.44) MAPTMAPK1LMNAKMT2AHPGD
SCHEMBL28381581 0.83 AKR1C3 (0.41) AKR1C3MAPTNPC1MAPK1HTT
SCHEMBL9747406 0.81 MAPT (0.37) AKR1C3MAPTNPC1MAPK1HTT
SCHEMBL9748692 0.81 KMT2A (0.39) AKR1C3MAPTNPC1MAPK1HTT
SCHEMBL10950202 0.73 GAA (0.34) AKR1C3MAPTNPC1HTTLMNA
SCHEMBL9747790 0.73 PGR (0.42) MAPTNPC1MAPK1HTTLMNA
SCHEMBL20939667 0.73 PDE7A (0.40) MAPK1HTTLMNA
SCHEMBL28424176 0.71 AKR1C3 (0.42) AKR1C3MAPTNPC1MAPK1HTT
SCHEMBL27970302 0.70 AKR1C3 (0.47) AKR1C3MAPTNPC1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221753-B1 TRANSDERMAL TREATMENT FOR PAIN AND INFLAMMATION WITH 2-AMINO-3-AROYLBENZENEACETIC ACIDS, SALTS AND ESTERS A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1992-01-08 EP disclosed
US-4683242-A Transdermal treatment for pain and inflammation with 2-amino-3-aroylbenzeneacetic acids, salts and esters A. H. ROBINS COMPANY, INCORPORATED (US) 1987-07-28 US disclosed
EP-0221753-A2 Transdermal treatment for pain and inflammation with 2-amino-3-aroylbenzeneacetic acids, salts and esters A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1987-05-13 EP disclosed