SCHEMBL9749314

SCHEMBL9749314

O=C(O)CSc1scnc1OC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 2/20 0.36
FFAR1 O14842 1/20 0.34
ALDH1A1 P00352 2/20 0.34
ALOX15 P16050 1/20 0.33
NOTUM Q6P988 3/20 0.33
MAP3K8 P41279 1/20 0.33
GAA P10253 2/20 0.33
KDM4E B2RXH2 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PHGDH O43175 1/20 0.32
CSNK2A2 P19784 3/20 0.32
CSNK2B P67870 3/20 0.32
CSNK2A1 P68400 3/20 0.32
PRNP P04156 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9748003 0.77 PTGS1 (0.36) HSD17B10CYP1A2KMT2AFFAR1ALDH1A1
SCHEMBL9750280 0.76 PTPRG (0.45) CYP1A2CYP2C19KMT2AALDH1A1GAA
SCHEMBL10688331 0.75 CYP1A2 (0.43) HSD17B10CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL9749147 0.73 MAPK1 (0.40) HSD17B10KMT2AFFAR1ALDH1A1ALOX15
SCHEMBL9852576 0.68 KDM4E (0.34) KDM4EL3MBTL1
SCHEMBL10872677 0.68 KDM4E (0.42) KDM4EL3MBTL1
SCHEMBL10432526 0.63 KDM4E (0.57) HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL10432894 0.60 KDM4E (0.35) CYP1A2CYP3A4KDM4E
SCHEMBL9706738 0.60 ALOX15 (0.49) HSD17B10CYP1A2KMT2AFFAR1ALDH1A1
SCHEMBL5632525 0.60 CYP1A2 (0.46) HSD17B10CYP1A2CYP3A4CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0194572-B1 HETEROCYCLIC SULFIDES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1992-01-02 EP disclosed
EP-0194572-A1 Heterocyclic sulfides, process for their preparation and Medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1986-09-17 EP disclosed