SCHEMBL9748003

SCHEMBL9748003

COC(=O)CCSc1scnc1OC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.36
KMT2A Q03164 5/20 0.35
CXCR1 P25024 1/20 0.35
CXCR2 P25025 1/20 0.35
ALDH1A1 P00352 5/20 0.34
MEN1 O00255 3/20 0.34
RAB9A P51151 1/20 0.34
HSD17B10 Q99714 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
GSTP1 P09211 1/20 0.34
GSTM2 P28161 1/20 0.34
FFAR1 O14842 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
ABL1 P00519 1/20 0.32
RIN1 Q13671 1/20 0.32
TSHR P16473 1/20 0.32
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852546 0.89 PTGS1 (0.36) PTGS1KMT2ACXCR1CXCR2ALDH1A1
SCHEMBL9748843 0.84 PTGS1 (0.38) PTGS1KMT2ACXCR1CXCR2ALDH1A1
SCHEMBL9852499 0.81 KMT2A (0.40) PTGS1KMT2ACXCR1CXCR2ALDH1A1
SCHEMBL9749314 0.77 HSD17B10 (0.40) KMT2AALDH1A1HSD17B10FFAR1HPGD
SCHEMBL9749147 0.75 MAPK1 (0.40) KMT2AALDH1A1MEN1HSD17B10MAPT
SCHEMBL10685641 0.73 PTGS1 (0.39) PTGS1KMT2ACXCR1CXCR2ALDH1A1
SCHEMBL9750280 0.72 PTPRG (0.45) KMT2AALDH1A1MEN1RAB9ALMNA
SCHEMBL9748133 0.71 HSD17B10 (0.32) ALDH1A1HSD17B10MAPTMAPK1HPGD
SCHEMBL15737155 0.69 KMT2A (0.43) PTGS1KMT2ACXCR1CXCR2ALDH1A1
SCHEMBL9627261 0.68 KDM4E (0.43) KMT2AALDH1A1MEN1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0194572-B1 HETEROCYCLIC SULFIDES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1992-01-02 EP disclosed
EP-0409055-A1 Cephalosporin derivatives and processes for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1991-01-23 EP disclosed
EP-0194572-A1 Heterocyclic sulfides, process for their preparation and Medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1986-09-17 EP disclosed