SCHEMBL9749382

SCHEMBL9749382

Cc1ncsc1SCC(CC(=O)O)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
PKM P14618 1/20 0.40
CPA1 P15085 2/20 0.35
CPB1 P15086 1/20 0.35
CPA3 P15088 1/20 0.35
CPB2 Q96IY4 1/20 0.35
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
FOLH1 Q04609 3/20 0.33
MAPK1 P28482 2/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
ACLY P53396 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9749609 0.86 KDM4E (0.38) KDM4EPKMCPA3FOLH1
SCHEMBL9749540 0.83 KDM4E (0.46) KDM4EPKMALDH1A1MEN1KMT2A
SCHEMBL9749243 0.72 CPA1 (0.36) KDM4ECPA1CPB1CPA3CPB2
SCHEMBL4236238 0.65 KDM4E (0.43) KDM4EPKMALDH1A1MEN1KMT2A
SCHEMBL2208741 0.62 KDM4E (0.52) KDM4EPKMALDH1A1MEN1KMT2A
SCHEMBL759475 0.62 CPA1 (0.49) KDM4ECPA1CPB1CPA3CPB2
SCHEMBL7814875 0.62 KDM4E (0.34) KDM4EPKMALDH1A1MEN1KMT2A
SCHEMBL8573240 0.61 CPB2 (0.53) CPA1CPB1CPA3CPB2FOLH1
SCHEMBL1279680 0.60 KDM4E (0.50) KDM4EPKMALDH1A1MEN1KMT2A
SCHEMBL7779172 0.60 ALDH1A1 (0.53) KDM4EPKMALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0194572-B1 HETEROCYCLIC SULFIDES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1992-01-02 EP disclosed
US-4762848-A IMMUNE SYSTEM STIMULANTS, CYTOSTATIC AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1988-08-09 US disclosed
EP-0194572-A1 Heterocyclic sulfides, process for their preparation and Medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1986-09-17 EP disclosed