SCHEMBL9750446

SCHEMBL9750446

C=C1N(C)c2c(OCc3ccc(C)cc3)cc(C)cc2C1(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
NPC1 O15118 5/20 0.36
RAB9A P51151 5/20 0.36
MAPT P10636 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
RECQL P46063 2/20 0.36
LMNA P02545 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
GAA P10253 1/20 0.35
HPGD P15428 3/20 0.34
NPY1R P25929 1/20 0.34
NPY2R P49146 1/20 0.34
MAOB P27338 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11019682 0.91 MAPT (0.40) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL9750080 0.85 ALDH1A1 (0.39) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL9750274 0.77 MAOB (0.43) NPC1RAB9AMAOBSMN1; SMN2CASP3
SCHEMBL11020994 0.73 MAPT (0.45) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL9750449 0.71 MAPT (0.40) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL4602669 0.71 MPI (0.38) MAPTKMT2AKDM4E
SCHEMBL9750009 0.68 CHRNA7 (0.46) ALDH1A1NPC1RAB9AMAPTHPGD
SCHEMBL9750098 0.66 MAOB (0.46) MAOBKMT2A
SCHEMBL9750191 0.64 PDK2 (0.39) ALDH1A1MAPTRECQLLMNAGAA
SCHEMBL5850441 0.63 MAPT (0.41) RAB9AMAPTKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120858-A Condensation of 2-methyleneindoline and formic acid in acetic anhydride MILES INC. (US) 1992-06-09 US disclosed
EP-0058863-B1 PROCESS FOR THE PREPARATION OF TRIMETHINE DYESTUFFS BAYER AG (DE) 1985-01-23 EP disclosed
US-4419511-A Process for the preparation of trimethine dyestuffs BAYER AKTIENGESELLSCHAFT (US) 1983-12-06 US disclosed
EP-0058863-A1 Process for the preparation of trimethine dyestuffs BAYER AG (DE) 1982-09-01 EP disclosed