SCHEMBL9750451

SCHEMBL9750451

C=C1N(C)c2c(Oc3cccc(C)c3)cccc2C1(C)C

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
GAA P10253 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.38
AR P10275 2/20 0.36
ACHE P22303 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 2/20 0.34
GRIA2 P42262 1/20 0.34
HTT P42858 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GFER P55789 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
THRB P10828 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9750033 0.81 ALDH1A1 (0.38) ALDH1A1GAAL3MBTL1LMNAHTT
SCHEMBL9750256 0.77 ALDH1A1 (0.35) ALDH1A1GAAL3MBTL1SMN1; SMN2LMNA
SCHEMBL9750191 0.73 PDK2 (0.39) ALDH1A1GAAL3MBTL1LMNANPSR1
SCHEMBL9750080 0.73 ALDH1A1 (0.39) ALDH1A1L3MBTL1SMN1; SMN2LMNAHTT
SCHEMBL4603103 0.72 MEN1 (0.37) ALDH1A1GAALMNAHTTTDP1
SCHEMBL9750259 0.69 MAPT (0.46) ALDH1A1GAAL3MBTL1TDP1KMT2A
SCHEMBL5541683 0.69 ALDH1A1 (0.64) ALDH1A1GAAL3MBTL1ARACHE
SCHEMBL9750447 0.67 PGR (0.33) ALDH1A1L3MBTL1SMN1; SMN2LMNATDP1
SCHEMBL11020994 0.67 MAPT (0.45) ALDH1A1GAAL3MBTL1SMN1; SMN2LMNA
SCHEMBL11019576 0.66 MAPT (0.46) ALDH1A1GAAL3MBTL1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120858-A Condensation of 2-methyleneindoline and formic acid in acetic anhydride MILES INC. (US) 1992-06-09 US disclosed
EP-0058863-B1 PROCESS FOR THE PREPARATION OF TRIMETHINE DYESTUFFS BAYER AG (DE) 1985-01-23 EP disclosed
US-4419511-A Process for the preparation of trimethine dyestuffs BAYER AKTIENGESELLSCHAFT (US) 1983-12-06 US disclosed
EP-0058863-A1 Process for the preparation of trimethine dyestuffs BAYER AG (DE) 1982-09-01 EP disclosed