SCHEMBL9751295

SCHEMBL9751295

O=C(Cl)SC1(c2ccccc2)N=NN=N1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.33
F2 P00734 1/20 0.33
AKR1C1 Q04828 1/20 0.32
CES2 O00748 3/20 0.32
CES1 P23141 3/20 0.32
ALDH1A1 P00352 1/20 0.32
KIF11 P52732 2/20 0.31
BCHE P06276 1/20 0.31
POLB P06746 1/20 0.31
APEX1 P27695 1/20 0.31
RECQL P46063 1/20 0.31
RAB9A P51151 1/20 0.31
BLM P54132 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
OPRM1 P35372 1/20 0.30
HSD11B1 P28845 1/20 0.30
HDAC4 P56524 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6385367 0.73 OPRM1 (0.30) OPRM1
SCHEMBL10872352 0.71 ALDH1A1 (0.41) ALDH1A1MEN1KMT2A
SCHEMBL11386287 0.71 ALDH1A1 (0.47) ALDH1A1OPRM1HDAC4
SCHEMBL10577287 0.70 OPRM1 (0.32) LMNAALDH1A1L3MBTL1OPRM1
SCHEMBL9751463 0.67 ALDH1A1 (0.36) LMNAF2AKR1C1ALDH1A1MEN1
SCHEMBL27746475 0.66 AKR1C1 (0.42) LMNAF2AKR1C1CES2CES1
SCHEMBL5168259 0.63 OPRM1 (0.38) LMNAAKR1C1CES2CES1ALDH1A1
SCHEMBL434296 0.62 KMT2A (0.33) AKR1C1ALDH1A1RAB9ABLMMEN1
SCHEMBL4666989 0.62 CYP2C9 (0.33) LMNAAKR1C1ALDH1A1BLMMEN1
SCHEMBL3819684 0.62 P2RX1 (0.33) RAB9AMEN1KMT2AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0396709-A4 HUMAN LEUKOCYTE ELASTASE INHIBITORS AND METHODS OF PRODUCING AND USING SAME 1991-05-22 EP disclosed
EP-0396709-A1 HUMAN LEUKOCYTE ELASTASE INHIBITORS AND METHODS OF PRODUCING AND USING SAME UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 1990-11-14 EP disclosed