SCHEMBL9753687

SCHEMBL9753687

COC(=O)c1ccc2c(C(C)C)c(C=O)c(-c3ccc(F)cc3)nn12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
HSD17B10 Q99714 2/20 0.39
GAA P10253 1/20 0.39
ALOX15 P16050 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
CYP3A4 P08684 1/20 0.36
GCGR P47871 1/20 0.35
PTGS2 P35354 2/20 0.35
HPGD P15428 1/20 0.34
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
KDM5B Q9UGL1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27438907 0.91 ALDH1A1 (0.37) ALDH1A1KDM4EHSD17B10GAAALOX15
SCHEMBL9753310 0.91 ALDH1A1 (0.37) ALDH1A1KDM4EHSD17B10GAAALOX15
SCHEMBL9753038 0.83 GCGR (0.47) ALDH1A1KDM4EHSD17B10GAAALOX15
SCHEMBL9753767 0.82 HMGCR (0.39) ALDH1A1CYP3A4HMGCR
SCHEMBL9753762 0.82 HMGCR (0.39) ALDH1A1CYP3A4HMGCR
SCHEMBL9753738 0.81 CACNA1F (0.42) KDM4EHSD17B10CA12CA1CA2
SCHEMBL9753740 0.81 CA12 (0.33) ALDH1A1KDM4EHSD17B10GAAALOX15
SCHEMBL9753096 0.81 HMGCR (0.51) ALDH1A1CYP2C9CYP3A4PTGS2HMGCR
SCHEMBL9752928 0.81 MAPK14 (0.43) ALDH1A1PTGS2KDM5B
SCHEMBL9753416 0.81 POLB (0.37) ALDH1A1PTGS2KDM5BHMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed