SCHEMBL9753740

SCHEMBL9753740

COC(=O)C1=C(C)N(c2ccc3c(C(C)C)c(C=O)c(-c4ccc(F)cc4)nn23)C(C)=C(C(=O)OC)C1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
ALDH1A1 P00352 6/20 0.32
MAPT P10636 3/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HMGCR P04035 1/20 0.31
KDM4E B2RXH2 3/20 0.31
HSD17B10 Q99714 2/20 0.31
PTGS2 P35354 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
GCGR P47871 1/20 0.31
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753687 0.81 ALDH1A1 (0.39) CA12CA1CA2CA9ALDH1A1
SCHEMBL9753738 0.75 CACNA1F (0.42) CA12CA1CA2CA9LMNA
SCHEMBL9752928 0.75 MAPK14 (0.43) ALDH1A1PTGS2KCNK3
SCHEMBL9753416 0.73 POLB (0.37) ALDH1A1HMGCRPTGS2KCNK3
SCHEMBL27438907 0.73 ALDH1A1 (0.37) CA12CA1CA2CA9ALDH1A1
SCHEMBL9753310 0.73 ALDH1A1 (0.37) CA12CA1CA2CA9ALDH1A1
SCHEMBL9753119 0.72 PTGS2 (0.36) ALDH1A1PTGS2KCNK3
SCHEMBL9753114 0.72 MAPK14 (0.42) ALDH1A1PTGS2
SCHEMBL9753314 0.71 KDM5B (0.34) ALDH1A1HMGCRPTGS2KCNK3
SCHEMBL9752970 0.71 KDM5B (0.34) ALDH1A1PTGS2KCNK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed