SCHEMBL9754290

SCHEMBL9754290

COc1ccc2cc(CCc3sc(-c4ccccc4)nc3O)ccc2c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.54
PTGDR2 Q9Y5Y4 3/20 0.48
TRPM8 Q7Z2W7 3/20 0.47
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAPT P10636 1/20 0.45
MAOA P21397 1/20 0.45
SLC6A2 P23975 1/20 0.45
RAB9A P51151 1/20 0.45
SLC6A3 Q01959 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PTGS1 P23219 1/20 0.44
AKR1C3 P42330 1/20 0.44
AKR1C2 P52895 1/20 0.44
CDC7 O00311 1/20 0.43
DBF4 Q9UBU7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754402 0.80 ALOX5 (0.56) ALOX5KDM4ENPC1LMNATP53
SCHEMBL9630221 0.78 TRPM8 (0.54) ALOX5PTGDR2TRPM8KDM4ECDC7
SCHEMBL9629404 0.74 TRPM8 (0.59) ALOX5TRPM8CDC7DBF4
SCHEMBL9754206 0.72 ALOX5 (0.53) ALOX5TRPM8NPC1LMNACYP1A2
SCHEMBL9630543 0.72 TRPM8 (0.57) ALOX5TRPM8CDC7DBF4
SCHEMBL9754018 0.71 ALOX5 (0.52) ALOX5TRPM8NPC1LMNACYP1A2
Potassium SCHEMBL9754024 0.71 ALOX5 (0.52) ALOX5TRPM8NPC1LMNACYP1A2
SCHEMBL9628554 0.71 TRPM8 (0.62) ALOX5PTGDR2TRPM8MAPTCDC7
SCHEMBL9629437 0.71 ALOX5 (1.00) ALOX5PTGDR2TRPM8KDM4ENPC1
SCHEMBL15662821 0.67 CYP1A2 (0.61) KDM4ENPC1LMNATP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991008744-A1 THIAZOLE LIPOXYGENASE-INHIBITING COMPOUNDS DERIVED FROM NON-STEROIDAL ANTIINFLAMMATORY CARBOXYLIC ACIDS ABBOTT LABORATORIES (US) 1991-06-27 WO disclosed