SCHEMBL9754402

SCHEMBL9754402

COc1ccc2cc(CCc3nc(O)c(-c4ccccc4)s3)ccc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.56
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
MAOA P21397 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
PTGS1 P23219 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754290 0.80 ALOX5 (0.54) ALOX5NPC1RAB9AKDM4ELMNA
SCHEMBL9754002 0.75 ALOX5 (0.47) ALOX5MEN1KMT2APTGS2
SCHEMBL9629437 0.72 ALOX5 (1.00) ALOX5NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL9754071 0.71 ALOX5 (0.53) ALOX5NPC1RAB9ALMNACYP1A2
SCHEMBL9630571 0.70 ALOX5 (0.53) ALOX5TP53MAPTSMN1; SMN2
SCHEMBL8358048 0.69 BCHE (0.55) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL9782162 0.69 PTGS2 (0.49) CYP1A2MAPTPTGS2
SCHEMBL9754030 0.68 ALOX5 (0.44) ALOX5MEN1KMT2APTGS2
Nabumetone SCHEMBL3362072 0.68 RAB9A (0.86) NPC1RAB9AKDM4ELMNATP53
SCHEMBL2663510 0.67 CYP1A2 (0.65) ALOX5NPC1RAB9AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991008744-A1 THIAZOLE LIPOXYGENASE-INHIBITING COMPOUNDS DERIVED FROM NON-STEROIDAL ANTIINFLAMMATORY CARBOXYLIC ACIDS ABBOTT LABORATORIES (US) 1991-06-27 WO disclosed