SCHEMBL9754611

SCHEMBL9754611

Cn1c2ccccc2c2sc3c(C=O)cccc3c21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
IMPDH2 P12268 1/20 0.44
ALKBH5 Q6P6C2 1/20 0.41
FTO Q9C0B1 1/20 0.41
LMNA P02545 3/20 0.40
GPR3 P46089 1/20 0.39
MAPT P10636 6/20 0.39
HTT P42858 6/20 0.39
NPSR1 Q6W5P4 5/20 0.39
HPGD P15428 3/20 0.39
AHR P35869 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
POLB P06746 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
KDM4E B2RXH2 4/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2786309 0.75 CYP2A6 (0.50) ALDH1A1IMPDH2LMNAHTTHPGD
SCHEMBL31689733 0.75 CYP2A6 (0.50) ALDH1A1IMPDH2LMNAHTTHPGD
SCHEMBL9754492 0.73 MAPT (0.49) ALDH1A1ALKBH5FTOLMNAGPR3
SCHEMBL9755646 0.71 GPR3 (0.52) ALDH1A1IMPDH2ALKBH5FTOLMNA
SCHEMBL9754575 0.71 ALDH1A1 (0.44) ALDH1A1IMPDH2ALKBH5FTOLMNA
SCHEMBL9754604 0.70 AHR (0.44) ALDH1A1IMPDH2ALKBH5FTOLMNA
SCHEMBL9779016 0.69 AHR (0.51) ALDH1A1IMPDH2ALKBH5FTOLMNA
SCHEMBL9754503 0.68 PTGER4 (0.43) ALDH1A1LMNAMAPTHTTHPGD
SCHEMBL30705823 0.67 CYP2A6 (0.48) ALDH1A1IMPDH2LMNAGPR3MAPT
SCHEMBL9525819 0.67 CYP2A6 (0.48) ALDH1A1IMPDH2LMNAGPR3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991014688-A1 HETERO POLYCYCLIC BIOCIDAL COMPOUNDS AND THEIR USE IN MEDECINE THE WELLCOME FOUNDATION LIMITED (GB) 1991-10-03 WO disclosed
EP-0447703-A1 Hetero polycyclic biocidal compounds, their synthesis and intermediates therefor,formulations containing them and their use in medicine THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-25 EP disclosed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed