SCHEMBL9756628

SCHEMBL9756628

COc1ccc(CC2C3CCCC=C3CCN2C)cc1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
HRH3 Q9Y5N1 3/20 0.40
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9441400 0.82 BCHE (0.40) BCHEACHEHRH3SIGMAR1
SCHEMBL11084149 0.70 BCHE (0.44) BCHEACHEHRH3SIGMAR1
SCHEMBL2066096 0.69 OPRK1 (0.43) HRH3SIGMAR1
SCHEMBL11760720 0.69 HRH3 (0.46) BCHEACHEHRH3SIGMAR1
SCHEMBL11768994 0.69 HRH3 (0.46) BCHEACHEHRH3SIGMAR1
SCHEMBL11769008 0.69 HRH3 (0.46) BCHEACHEHRH3SIGMAR1
SCHEMBL11760698 0.69 HRH3 (0.46) BCHEACHEHRH3SIGMAR1
SCHEMBL11760710 0.69 HRH3 (0.46) BCHEACHEHRH3SIGMAR1
SCHEMBL2066095 0.69 BCHE (0.44) BCHEACHEHRH3SIGMAR1
SCHEMBL11766646 0.68 HRH3 (0.45) BCHEACHEHRH3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283848-B1 PROCESS FOR THE PREPARATION OF ISOQUINOLINES F. HOFFMANN-LA ROCHE AG (CH) 1991-05-15 EP disclosed
EP-0283848-A1 Process for the preparation of isoquinolines F. HOFFMANN-LA ROCHE AG (CH) 1988-09-28 EP disclosed