SCHEMBL9757224

SCHEMBL9757224

C=C(c1ccc(COc2ccc3sc(C(=O)O)c(C)c3c2)cc1)c1ccc2ccccc2n1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.48
CYSLTR1 Q9Y271 5/20 0.44
PDE10A Q9Y233 1/20 0.42
GPBAR1 Q8TDU6 2/20 0.41
SCD O00767 1/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
TBXAS1 P24557 1/20 0.38
ALOX5 P09917 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757147 0.90 EDNRA (0.42) EDNRANPC1TBXAS1
SCHEMBL9757054 0.85 PDE10A (0.58) EDNRACYSLTR1PDE10AGPBAR1ALOX5
SCHEMBL9757226 0.82 EDNRA (0.48) EDNRACYSLTR1PDE10ANPC1MAPT
SCHEMBL9757227 0.82 EDNRA (0.48) EDNRACYSLTR1PDE10ANPC1MAPT
SCHEMBL9757151 0.81 NR4A2 (0.43) EDNRACYSLTR1GPBAR1TBXAS1
SCHEMBL9757076 0.80 ALOX5 (0.59) EDNRACYSLTR1PDE10AGPBAR1ALOX5
SCHEMBL9757119 0.77 PDE10A (0.54) CYSLTR1PDE10AGPBAR1ALOX5
SCHEMBL9757233 0.76 CYSLTR1 (0.55) CYSLTR1PDE10AGPBAR1ALOX5
SCHEMBL9757716 0.74 ALOX5AP (0.48) EDNRACYSLTR1PDE10AALOX5
SCHEMBL9757124 0.72 ALOX5 (0.58) CYSLTR1PDE10AGPBAR1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed