SCHEMBL9757147

SCHEMBL9757147

C=C(c1ccc(COc2ccc3sc(C(=O)O)c(C)c3c2)cc1)c1ccc2ccc(Cl)cc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.42
SLC26A4 O43511 1/20 0.40
KMT2A Q03164 1/20 0.40
NR4A2 P43354 2/20 0.39
RXRA P19793 2/20 0.39
RXRB P28702 2/20 0.39
RXRG P48443 2/20 0.39
TBXAS1 P24557 2/20 0.37
ALOX5AP P20292 2/20 0.37
CYP3A4 P08684 1/20 0.37
KCNH2 Q12809 1/20 0.37
MAOB P27338 3/20 0.36
MAOA P21397 2/20 0.36
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
BCL2 P10415 1/20 0.35
BCL2L1 Q07817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757224 0.90 EDNRA (0.48) EDNRATBXAS1NPC1
SCHEMBL9757151 0.90 NR4A2 (0.43) EDNRANR4A2RXRARXRBRXRG
SCHEMBL9757716 0.85 ALOX5AP (0.48) EDNRASLC26A4KMT2AALOX5APCYP3A4
SCHEMBL9757150 0.82 CYSLTR1 (0.43) EDNRASLC26A4KMT2ATBXAS1ALOX5AP
SCHEMBL9757075 0.81 ROCK1 (0.32) SLC26A4KMT2AALOX5APCYP3A4KCNH2
SCHEMBL9757206 0.79 NR4A2 (0.42) KMT2ANR4A2RXRARXRBRXRG
SCHEMBL9757078 0.75 CYSLTR1 (0.53)
SCHEMBL9757054 0.74 PDE10A (0.58) EDNRAALOX5AP
SCHEMBL9757226 0.72 EDNRA (0.48) EDNRAKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL9757227 0.72 EDNRA (0.48) EDNRAKMT2ANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed