SCHEMBL9759954

SCHEMBL9759954

CC(CO)N1c2ccccc2Sc2cccc(C#N)c21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.40
PTGS2 P35354 2/20 0.40
NOX1 Q9Y5S8 1/20 0.37
BCHE P06276 6/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
CYP2D6 P10635 3/20 0.36
LMNA P02545 2/20 0.36
CYP1A2 P05177 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SLC22A1 O15245 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ESR1 P03372 1/20 0.36
PRNP P04156 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
HTR1A P08908 1/20 0.36
CHRM5 P08912 1/20 0.36
ADRA2A P08913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9759522 0.86 PTGS1 (0.37) PTGS1PTGS2BCHEFNTAFNTB
SCHEMBL9759527 0.86 PTGS1 (0.37) PTGS1PTGS2BCHEFNTAFNTB
SCHEMBL9759957 0.82 PTGS1 (0.40) PTGS1PTGS2NOX1BCHEFNTA
SCHEMBL20345839 0.80 PTGS1 (0.54) PTGS1PTGS2NOX1BCHECYP2D6
SCHEMBL9331439 0.77 LMNA (0.46) PTGS1PTGS2BCHECYP2D6LMNA
SCHEMBL9331442 0.77 LMNA (0.46) PTGS1PTGS2BCHECYP2D6LMNA
SCHEMBL9791007 0.68 MAOA (0.48) PTGS1PTGS2NOX1BCHECYP2D6
SCHEMBL12386881 0.66 PTGS1 (0.51) PTGS1PTGS2BCHECYP2D6LMNA
SCHEMBL9331947 0.66 LMNA (0.41) PTGS1PTGS2NOX1BCHECYP2D6
SCHEMBL29960525 0.66 MAOA (0.34) NOX1BCHEFNTAFNTBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5049669-A Also diuretics RHONE-POULENC SANTE (FR) 1991-09-17 US disclosed
US-4985419-A Analgesics, Diuretics RHONE-POULENC SANTE (FR) 1991-01-15 US disclosed
US-4912105-A Derivatives of phenothiazine and the compositions which contain them RHONE-POULENC SANTE (FR) 1990-03-27 US disclosed