SCHEMBL9759957

SCHEMBL9759957

CCC(O)N1c2ccccc2Sc2cccc(C#N)c21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.40
PTGS2 P35354 2/20 0.40
BCHE P06276 9/20 0.38
MAPT P10636 3/20 0.38
NOX1 Q9Y5S8 1/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
CYP2D6 P10635 2/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
GAA P10253 1/20 0.35
POLB P06746 1/20 0.35
ATM Q13315 1/20 0.35
ACHE P22303 3/20 0.35
MAOA P21397 2/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
ALOX15 P16050 2/20 0.35
ALOX12 P18054 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9759954 0.82 PTGS1 (0.40) PTGS1PTGS2BCHEMAPTNOX1
SCHEMBL9759522 0.79 PTGS1 (0.37) PTGS1PTGS2BCHEMAPTFNTA
SCHEMBL9759527 0.79 PTGS1 (0.37) PTGS1PTGS2BCHEMAPTFNTA
SCHEMBL9331534 0.77 LMNA (0.46) PTGS1PTGS2BCHEMAPTCYP2D6
SCHEMBL4595129 0.68 MAOA (0.48) PTGS1PTGS2BCHEMAPTCYP2D6
SCHEMBL12386881 0.66 PTGS1 (0.51) PTGS1PTGS2BCHEMAPTCYP2D6
SCHEMBL29960525 0.66 MAOA (0.34) BCHEMAPTNOX1FNTAFNTB
SCHEMBL8142099 0.65 PTGS1 (0.59) PTGS1PTGS2BCHEMAPTNOX1
SCHEMBL23954417 0.65 MAOA (0.38) NOX1TSHRMAOAKDM4EALDH1A1
SCHEMBL28842814 0.65 KDM4E (0.36) BCHEMAPTNOX1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5049669-A Also diuretics RHONE-POULENC SANTE (FR) 1991-09-17 US disclosed
US-4985419-A Analgesics, Diuretics RHONE-POULENC SANTE (FR) 1991-01-15 US disclosed