SCHEMBL9760930

SCHEMBL9760930

Cn1c(=O)[nH]c2ccc(C(=O)c3ccccc3)cc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.56
ADORA2B P29275 2/20 0.56
ADORA2A P29274 1/20 0.56
ADORA1 P30542 1/20 0.56
ALDH1A1 P00352 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
GLA P06280 1/20 0.50
HPGD P15428 3/20 0.46
BRD4 O60885 1/20 0.44
POLB P06746 1/20 0.44
RAB9A P51151 1/20 0.44
PARG Q86W56 1/20 0.43
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
ATM Q13315 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CNR2 P34972 1/20 0.41
HTR3A P46098 1/20 0.41
LMNA P02545 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9761035 0.80 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2HPGDPOLBTDP1
SCHEMBL2115896 0.79 KDM4E (0.58) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL2116094 0.79 HTR3A (0.50) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL14927289 0.77 ADORA3 (0.43) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL4550112 0.76 HTR3A (0.47) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL14927286 0.75 ADORA3 (0.41) ADORA3ADORA2BADORA2AADORA1GLA
SCHEMBL11069044 0.74 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2HPGDRAB9AATM
SCHEMBL9759896 0.74 CA12 (0.51) ALDH1A1SMN1; SMN2HPGDBRD4POLB
SCHEMBL4252129 0.74 KDM4E (0.64) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL29897963 0.73 ADORA3 (1.00) ADORA3ADORA2BADORA2AADORA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037829-A Antitumor Activity; Androgen, Estrogen Inhibitors; Suppress The Plasma Elimination Of Retinoids JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-06 US disclosed