SCHEMBL9764104

SCHEMBL9764104

COc1ccc(-n2c(-c3ccccc3)c(-c3ccc(F)cc3)c(C=O)c2C(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
OXTR P30559 1/20 0.38
SRC P12931 1/20 0.38
BRAF P15056 1/20 0.38
KDR P35968 1/20 0.38
GLA P06280 2/20 0.37
MDM4 O15151 1/20 0.37
MDM2 Q00987 1/20 0.37
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GBA1 P04062 1/20 0.36
NLRP3 Q96P20 1/20 0.35
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764185 0.90 KDM4E (0.48) ALDH1A1KDM4ETDP1L3MBTL1CYP3A4
SCHEMBL9764095 0.78 ALDH1A1 (0.43) ALDH1A1KDM4ETDP1L3MBTL1PTGS2
SCHEMBL9658354 0.77 ALDH1A1 (0.41) ALDH1A1KDM4ETDP1L3MBTL1PTGS2
SCHEMBL9518289 0.77 HMGCR (0.47) ALDH1A1KDM4ETDP1L3MBTL1MEN1
SCHEMBL12758829 0.73 ALDH1A1 (0.44) ALDH1A1KDM4ETDP1L3MBTL1NPSR1
SCHEMBL9764313 0.72 PTGS2 (0.43) ALDH1A1KDM4ETDP1L3MBTL1PTGS2
SCHEMBL13302194 0.72 HMGCR (0.44) ALDH1A1KDM4ETDP1L3MBTL1CYP3A4
SCHEMBL13302361 0.72 HMGCR (0.42) ALDH1A1KDM4ETDP1L3MBTL1CYP3A4
SCHEMBL9024278 0.69 PTGS2 (0.38) ALDH1A1PTGS1PTGS2
SCHEMBL9764105 0.68 MEN1 (0.39) ALDH1A1KDM4ETDP1L3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032590-A Substituted hydroxylamines BAYER AKTIENGESELLSCHAFT (DE) 1991-07-16 US disclosed
US-4994462-A N,N-Bis(nipecotyl)piperazines RESEARCH CORPORATION (US) 1991-02-19 US disclosed
US-4968681-A Substituted hydroxylamines BAYER AKTIENGESELLSCHAFT (DE) 1990-11-06 US disclosed
EP-0317845-A2 Substituted hydroxyl amines BAYER AG (DE) 1989-05-31 EP disclosed