SCHEMBL9764301

SCHEMBL9764301

COc1ccc(CCCOCCCCCN(Cc2ccccc2)CC(O)c2cc(Cl)c(N)c(Cl)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 3/20 0.45
L3MBTL1 Q9Y468 3/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
ADRB2 P07550 1/20 0.38
BCHE P06276 2/20 0.38
ALOX5 P09917 1/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
MEP1B Q16820 1/20 0.37
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764694 0.96 NR1H3 (0.45) NR1H3L3MBTL1TDP1MAOAMAOB
SCHEMBL9764371 0.91 ADRB2 (0.41) NR1H3ADRB2BCHETSHRKCNH2
SCHEMBL9764429 0.89 ADRB2 (0.41) NR1H3MAOBADRB2BCHETSHR
SCHEMBL9764456 0.89 ADRB2 (0.41) NR1H3MAOBADRB2BCHETSHR
SCHEMBL10346955 0.89 TDP1 (0.52) NR1H3L3MBTL1TDP1MAOAMAOB
SCHEMBL10389958 0.88 ADRB2 (0.41) NR1H3TDP1ADRB2BCHETSHR
SCHEMBL9764389 0.88 ADRB2 (0.39) NR1H3ADRB2BCHEKCNH2
SCHEMBL10417482 0.88 SLC2A1 (0.39) NR1H3ADRB2BCHETSHRKCNH2
SCHEMBL9324009 0.87 MAOB (0.39) NR1H3MAOAMAOBBCHE
SCHEMBL9321535 0.86 MAOB (0.37) NR1H3MAOAMAOBADRB2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed